NCI-H2228 · CELL-LINE · Homo sapiens
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NCI-H2228
Review this target as NCI-H2228.
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This review treats NCI-H2228 as ChEMBL target CHEMBL1075536. Disease framing currently uses the Open Targets-ready proxy contract.
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| Preferred Name | NCI-H2228 |
| Target Type | CELL-LINE |
| Organism | Homo sapiens |
Reviewable protein naming and mapping context for this target snapshot.
Review this target as NCI-H2228.
| ChEMBL ID | pChEMBL | Type | Value (nM) | Phase |
|---|---|---|---|---|
| CHEMBL5270787 | 9.52 | IC50 | 0.3 | Preclinical |
| CHEMBL888 | 9.5 | IC50 | 0.314 | Approved |
| CHEMBL94657 | 9.32 | IC50 | 0.4727 | Clinical |
| CHEMBL105 | 9.1 | IC50 | 0.7963 | Approved |
| CHEMBL3128069 | 9.1 | IC50 | 0.8 | Preclinical |
| CHEMBL1738797 | 8.19 | IC50 | 6.5 | Approved |
| CHEMBL3545252 | 8.14 | IC50 | 7.253 | Approved |
| CHEMBL96926 | 8.1 | IC50 | 8.004 | Preclinical |
| CHEMBL4474454 | 8.0 | IC50 | 10.0 | Preclinical |
| CHEMBL252164 | 7.97 | IC50 | 10.64 | Clinical |
| BAO Format | Assays | Compounds | Avg pChEMBL |
|---|---|---|---|
| cell-based format | 225 | 684 | 6.2 |
| organism-based format | 49 | 0 | — |