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Assay Detail

CHEMBL1004216

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Vaccinia virus Copenhagen in HFF cells assessed as reduction plaque formation after 3 days
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Vaccinia virus
Cell Type HFF
Confidence 1 — Organism
Curated By Autocuration

Target

Vaccinia virus (CHEMBL613493)
Type ORGANISM
Organism Vaccinia virus

Publication

Synergistic efficacy of the combination of ST-246 with CMX001 against orthopoxviruses.
Quenelle DC, Prichard MN, Keith KA, Hruby DE, Jordan R, Painter GR, Robertson A, Kern ER.
Antimicrob Agents Chemother (2007) 51 : 4118 -4124
PubMed 17724153 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 3 6.23 7.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1257073 TECOVIRIMAT 4.0 1 7.30
CHEMBL203321 BRINCIDOFOVIR 4.0 1 6.85
CHEMBL5314375 CIDOFOVIR 4.0 1 4.54

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1257073 TECOVIRIMAT EC50 = 50.0 nM 7.30
CHEMBL203321 BRINCIDOFOVIR EC50 = 140.0 nM 6.85
CHEMBL5314375 CIDOFOVIR EC50 = 29200.0 nM 4.54