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Assay Detail

CHEMBL1006052

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human HL60
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HL-60
Confidence 1 — Organism
Curated By Autocuration

Target

HL-60 (CHEMBL383)
Type CELL-LINE
Organism Homo sapiens

Publication

A labdane diterpene glucoside from the rhizomes of Curcuma mangga.
Abas F, Lajis NH, Shaari K, Israf DA, Stanslas J, Yusuf UK, Raof SM.
J Nat Prod (2005) 68 : 1090 -1093
PubMed 16038556 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 4.71 5.14

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL512317 ZERUMIN B 1 5.14
CHEMBL179512 DEMETHOXYCURCUMIN 1 4.62
CHEMBL105350 BISDEMETHOXYCURCUMIN 1 4.60
CHEMBL140 CURCUMIN 3.0 1 4.47
CHEMBL71851 SCOPOLETIN 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL512317 ZERUMIN B IC50 = 7210.0 nM 5.14
CHEMBL179512 DEMETHOXYCURCUMIN IC50 = 24210.0 nM 4.62
CHEMBL105350 BISDEMETHOXYCURCUMIN IC50 = 25120.0 nM 4.60
CHEMBL140 CURCUMIN IC50 = 34220.0 nM 4.47
CHEMBL71851 SCOPOLETIN IC50 > 50000.0 nM -