Assay Detail
Binding
CHEMBL1007619
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Inhibition of bovine liver beta-galactosidase by spectrophotometry
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bos taurus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Glycosidase-inhibiting pyrrolidines and pyrrolizidines with a long side chain in Scilla peruviana.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 7 | 6.21 | 7.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL469435 | — | — | 1 | 7.05 |
| CHEMBL456077 | — | — | 1 | 5.36 |
| CHEMBL449851 | — | — | 1 | - |
| CHEMBL511823 | — | — | 1 | - |
| CHEMBL512479 | — | — | 1 | - |
| CHEMBL498968 | — | — | 1 | - |
| CHEMBL469437 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL469435 | — | IC50 | = | 90.0 | nM | 7.05 |
| CHEMBL456077 | — | IC50 | = | 4400.0 | nM | 5.36 |
| CHEMBL449851 | — | IC50 | = | 260000.0 | nM | - |
| CHEMBL511823 | — | IC50 | = | 130000.0 | nM | - |
| CHEMBL512479 | — | IC50 | = | 320000.0 | nM | - |
| CHEMBL498968 | — | IC50 | = | 830000.0 | nM | - |
| CHEMBL469437 | — | IC50 | = | 920000.0 | nM | - |