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Compound Detail

CHEMBL449851

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CC(O)C[C@H]1N[C@H](CO)[C@@H](O)[C@@H]1O

Basic Information

ChEMBL ID CHEMBL449851
Phase Preclinical
Structure Type MOL
InChI Key SKCBFFYDHKQEQU-NMBMWNOXSA-N
1
Targets
5
Activities
1
Assay Types
0
PK Parameters
7
Publications
0
Known Names

Molecular Properties

191.2
MW (Da)
-2.19
ALogP
5
HBA
5
HBD
93.0
PSA (Ų)
0.35
QED
0
Ro5 Violations
3
Rot. Bonds

Drug Information

Molecule Type Small molecule
Availability Unknown
Chirality Unknown

Flags

Natural Product First in Class Prodrug

Extended Properties

Molecular Formula C8H17NO4
MW 191.23
Aromatic Rings 0
Heavy Atoms 13
NP-Likeness 2.42

Activity Summary

IC50 5 meas. best 4.0

Target Activity Profile

Target Type Best pChEMBL Mean pChEMBL Best (nM) # Data
Unchecked
CHEMBL612545
IC50 4.0 4.0 100000.0 1

Activity Data Samples

Top measurements by pChEMBL value

Target Type Rel. Value Units pChEMBL Assay PubMed
Unchecked IC50 = 100000.0 nM 4.0 Inhibition of yeast alpha-glucosidase by spectrophotometry 15165148

Literature References

PubMed DOI Target Context # Activities
15165148 10.1021/np0499721 Unchecked 7
15165148 10.1021/np0499721 Beta-galactosidase 1
15165148 10.1021/np0499721 Beta-mannosidase 1
15165148 10.1021/np0499721 Tissue alpha-L-fucosidase 1
15165148 10.1021/np0499721 Acidic alpha-glucosidase 1
15165148 10.1021/np0499721 Lysosomal acid glucosylceramidase 1
15165148 10.1021/np0499721 Alpha-galactosidase 1

Data from ChEMBL 36 via Core Engine