Assay Detail
Binding
CHEMBL1009870
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to CB2 receptor
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Discovery of novel CB2 receptor ligands by a pharmacophore-based virtual screening workflow.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 8.00 | 8.47 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL371214 | — | — | 1 | 8.47 |
| CHEMBL498767 | — | — | 1 | 8.14 |
| CHEMBL73711 | — | — | 1 | 7.92 |
| CHEMBL408430 | — | — | 1 | 7.82 |
| CHEMBL497392 | — | — | 1 | 7.64 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL371214 | — | Ki | = | 3.4 | nM | 8.47 |
| CHEMBL498767 | — | Ki | = | 7.2 | nM | 8.14 |
| CHEMBL73711 | — | Ki | = | 12.0 | nM | 7.92 |
| CHEMBL408430 | — | Ki | = | 15.1 | nM | 7.82 |
| CHEMBL497392 | — | Ki | = | 22.7 | nM | 7.64 |