Assay Detail
Binding
CHEMBL1013161
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Inhibition of GST fused human recombinant ALK5 expressed in Sf9 cells by radioisotopic protein kinase assay
35
Total Activities
35
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | Sf9 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Synthesis and biological evaluation of trisubstituted imidazole derivatives as inhibitors of p38alpha mitogen-activated protein kinase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 35 | 7.44 | 7.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL492634 | — | — | 1 | 7.44 |
| CHEMBL495301 | — | — | 1 | - |
| CHEMBL480945 | — | — | 1 | - |
| CHEMBL480933 | — | — | 1 | - |
| CHEMBL481338 | — | — | 1 | - |
| CHEMBL519294 | — | — | 1 | - |
| CHEMBL481752 | — | — | 1 | - |
| CHEMBL520437 | — | — | 1 | - |
| CHEMBL480787 | — | — | 1 | - |
| CHEMBL481761 | — | — | 1 | - |
| CHEMBL519620 | — | — | 1 | - |
| CHEMBL479987 | — | — | 1 | - |
| CHEMBL492848 | — | — | 1 | - |
| CHEMBL480940 | — | — | 1 | - |
| CHEMBL492849 | — | — | 1 | - |
| CHEMBL493055 | — | — | 1 | - |
| CHEMBL522003 | — | — | 1 | - |
| CHEMBL493685 | — | — | 1 | - |
| CHEMBL493686 | — | — | 1 | - |
| CHEMBL492858 | — | — | 1 | - |
| CHEMBL480936 | — | — | 1 | - |
| CHEMBL481339 | — | — | 1 | - |
| CHEMBL481757 | — | — | 1 | - |
| CHEMBL481917 | — | — | 1 | - |
| CHEMBL481764 | — | — | 1 | - |
| CHEMBL482129 | — | — | 1 | - |
| CHEMBL520949 | — | — | 1 | - |
| CHEMBL482300 | — | — | 1 | - |
| CHEMBL482301 | — | — | 1 | - |
| CHEMBL520919 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL492634 | — | IC50 | = | 36.0 | nM | 7.44 |
| CHEMBL519294 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL492848 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL479987 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL519620 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL481761 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL480787 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL520437 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL481752 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL492849 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL481338 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL480933 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL480945 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL480944 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL521424 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL481354 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL481347 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL481513 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL481339 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL520919 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL482301 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL482300 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL520949 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL482129 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL481764 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL481917 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL481757 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL480940 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL480936 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL492858 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL493686 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL493685 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL522003 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL495301 | — | IC50 | > | 1000.0 | nM | - |
| CHEMBL493055 | — | IC50 | > | 1000.0 | nM | - |