Assay Detail
Binding
CHEMBL1013936
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]AF-DX384 from muscarinic M2 receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
The role of receptor binding in drug discovery.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 9.22 | 9.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL500996 | METHOCTRAMINE HYDROCHLORIDE | — | 1 | 9.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL500996 | METHOCTRAMINE HYDROCHLORIDE | Ki | = | 0.6 | nM | 9.22 |