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Assay Detail

CHEMBL1015213

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Inhibition of CYP3A1/CYP3A2-catalyzed erythromycin N-demethylase activity in dexamethasone-treated Sprague-Dawley rat liver microsomes by spectrophotometry
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Rattus norvegicus
Tissue Liver
Subcellular Microsome
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cytochrome P450 3A1 (CHEMBL3323)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Synthesis and evaluation of imidazole-dioxolane compounds as selective heme oxygenase inhibitors: effect of substituents at the 4-position of the dioxolane ring.
Vlahakis JZ, Hum M, Rahman MN, Jia Z, Nakatsu K, Szarek WA.
Bioorg Med Chem (2009) 17 : 2461 -2475
PubMed 19268600 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 11 5.55 5.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL208047 1 5.85
CHEMBL472975 1 5.75
CHEMBL475163 1 5.70
CHEMBL473375 1 5.70
CHEMBL515086 1 5.68
CHEMBL447959 1 5.66
CHEMBL473364 1 5.55
CHEMBL516064 1 5.47
CHEMBL464300 1 5.40
CHEMBL3216038 1 5.16
CHEMBL474379 1 5.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL208047 IC50 = 1400.0 nM 5.85
CHEMBL472975 IC50 = 1800.0 nM 5.75
CHEMBL475163 IC50 = 2000.0 nM 5.70
CHEMBL473375 IC50 = 2000.0 nM 5.70
CHEMBL515086 IC50 = 2100.0 nM 5.68
CHEMBL447959 IC50 = 2200.0 nM 5.66
CHEMBL473364 IC50 = 2800.0 nM 5.55
CHEMBL516064 IC50 = 3400.0 nM 5.47
CHEMBL464300 IC50 = 4000.0 nM 5.40
CHEMBL3216038 IC50 = 7000.0 nM 5.16
CHEMBL474379 IC50 = 6900.0 nM 5.16