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Assay Detail

CHEMBL1016594

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]LTD4 from LTD4 receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Intermediate

Target

Cysteinyl leukotriene receptor 1 (CHEMBL1798)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

The role of receptor binding in drug discovery.
Sweetnam PM, Caldwell L, Lancaster J, Bauer C, McMillan B, Kinnier WJ, Price CH.
J Nat Prod (1993) 56 : 441 -455
PubMed 8496700 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 9.22 9.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL288943 LEUKOTRIENE D4 -1.0 1 9.22

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL288943 LEUKOTRIENE D4 Ki = 0.6 nM 9.22