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Assay Detail

CHEMBL1017828

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against HIV1 in human MT2 cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human immunodeficiency virus 1
Cell Type MT2
Confidence 1 — Organism
Curated By Autocuration

Target

Human immunodeficiency virus 1 (CHEMBL378)
Type ORGANISM
Organism Human immunodeficiency virus 1

Publication

Evaluation of hexadecyloxypropyl-9-R-[2-(Phosphonomethoxy)propyl]- adenine, CMX157, as a potential treatment for human immunodeficiency virus type 1 and hepatitis B virus infections.
Painter GR, Almond MR, Trost LC, Lampert BM, Neyts J, De Clercq E, Korba BE, Aldern KA, Beadle JR, Hostetler KY.
Antimicrob Agents Chemother (2007) 51 : 3505 -3509
PubMed 17646420 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 10.70 10.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL473586 1 10.70
CHEMBL502317 1 10.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL473586 EC50 = 0.02 nM 10.70
CHEMBL502317 EC50 = 0.02 nM 10.70