Assay Detail
Functional
CHEMBL1024330
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antiviral activity against HIV isolate 584.000 030 by replication assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Human immunodeficiency virus |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Target
Human immunodeficiency virus (CHEMBL613758) ↗| Type | ORGANISM |
| Organism | Human immunodeficiency virus |
Publication
Heterobiaryl human immunodeficiency virus entry inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 7.65 | 7.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL549336 | — | — | 1 | 7.89 |
| CHEMBL337301 | — | — | 1 | 7.54 |
| CHEMBL238103 | — | — | 1 | 7.52 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL549336 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL337301 | — | IC50 | = | 29.0 | nM | 7.54 |
| CHEMBL238103 | — | IC50 | = | 30.0 | nM | 7.52 |