Assay Detail
Binding
CHEMBL1029934
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Inhibition of Huntingtin protein aggregation by cell based assay
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Intermediate |
Publication
Potent inhibitors of Huntingtin protein aggregation in a cell-based assay.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 29 | 5.50 | 6.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL493153 | — | — | 1 | 6.15 |
| CHEMBL493327 | — | — | 1 | 5.97 |
| CHEMBL500972 | — | — | 1 | 5.96 |
| CHEMBL495005 | — | — | 1 | 5.88 |
| CHEMBL494838 | — | — | 1 | 5.66 |
| CHEMBL509988 | — | — | 1 | 5.56 |
| CHEMBL149800 | — | — | 1 | 5.46 |
| CHEMBL445226 | — | — | 1 | 5.44 |
| CHEMBL494130 | — | — | 1 | 5.35 |
| CHEMBL444229 | — | — | 1 | 5.28 |
| CHEMBL494325 | — | — | 1 | 5.27 |
| CHEMBL494326 | — | — | 1 | 5.21 |
| CHEMBL493348 | — | — | 1 | 5.20 |
| CHEMBL449571 | — | — | 1 | 5.09 |
| CHEMBL153483 | — | — | 1 | 4.98 |
| CHEMBL451222 | — | — | 1 | - |
| CHEMBL493324 | — | — | 1 | - |
| CHEMBL489053 | — | — | 1 | - |
| CHEMBL506969 | — | — | 1 | - |
| CHEMBL442675 | — | — | 1 | - |
| CHEMBL493349 | — | — | 1 | - |
| CHEMBL493350 | — | — | 1 | - |
| CHEMBL493325 | — | — | 1 | - |
| CHEMBL153733 | — | — | 1 | - |
| CHEMBL450176 | — | — | 1 | - |
| CHEMBL493308 | — | — | 1 | - |
| CHEMBL522502 | — | — | 1 | - |
| CHEMBL493309 | — | — | 1 | - |
| CHEMBL494129 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL493153 | — | IC50 | = | 710.0 | nM | 6.15 |
| CHEMBL493327 | — | IC50 | = | 1070.0 | nM | 5.97 |
| CHEMBL500972 | — | IC50 | = | 1110.0 | nM | 5.96 |
| CHEMBL495005 | — | IC50 | = | 1310.0 | nM | 5.88 |
| CHEMBL494838 | — | IC50 | = | 2210.0 | nM | 5.66 |
| CHEMBL509988 | — | IC50 | = | 2740.0 | nM | 5.56 |
| CHEMBL149800 | — | IC50 | = | 3440.0 | nM | 5.46 |
| CHEMBL445226 | — | IC50 | = | 3630.0 | nM | 5.44 |
| CHEMBL494130 | — | IC50 | = | 4480.0 | nM | 5.35 |
| CHEMBL444229 | — | IC50 | = | 5260.0 | nM | 5.28 |
| CHEMBL494325 | — | IC50 | = | 5360.0 | nM | 5.27 |
| CHEMBL494326 | — | IC50 | = | 6130.0 | nM | 5.21 |
| CHEMBL493348 | — | IC50 | = | 6380.0 | nM | 5.20 |
| CHEMBL449571 | — | IC50 | = | 8130.0 | nM | 5.09 |
| CHEMBL153483 | — | IC50 | = | 10500.0 | nM | 4.98 |
| CHEMBL451222 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL493324 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL489053 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL506969 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL442675 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL493349 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL493350 | — | IC50 | > | 15800.0 | nM | - |
| CHEMBL493325 | — | IC50 | - | — | - | |
| CHEMBL153733 | — | IC50 | - | — | - | |
| CHEMBL450176 | — | IC50 | - | — | - | |
| CHEMBL493308 | — | IC50 | - | — | - | |
| CHEMBL522502 | — | IC50 | - | — | - | |
| CHEMBL493309 | — | IC50 | - | — | - | |
| CHEMBL494129 | — | IC50 | - | — | - |