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Assay Detail

CHEMBL1029935

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Binding
Inhibition of Huntingtin protein aggregation by yeast based assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Intermediate

Target

Huntingtin (CHEMBL5514)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Potent inhibitors of Huntingtin protein aggregation in a cell-based assay.
Rinderspacher A, Cremona ML, Liu Y, Deng SX, Xie Y, Gong G, Aulner N, Többen U, Myers K, Chung C, Andersen M, Vidović D, Schürer S, Brandén L, Yamamoto A, Landry DW.
Bioorg Med Chem Lett (2009) 19 : 1715 -1717
PubMed 19243939 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 3 4.30 4.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL449571 1 4.30
CHEMBL494325 1 4.30
CHEMBL494326 1 4.30

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL449571 EC50 = 50000.0 nM 4.30
CHEMBL494325 EC50 = 50000.0 nM 4.30
CHEMBL494326 EC50 = 50000.0 nM 4.30