Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL1034009

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against influenza H2N2 virus
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism H2N2 subtype
Confidence 1 — Organism
Curated By Autocuration

Target

H2N2 subtype (CHEMBL612765)
Type ORGANISM
Organism H2N2 subtype

Publication

Unified QSAR approach to antimicrobials. 4. Multi-target QSAR modeling and comparative multi-distance study of the giant components of antiviral drug-drug complex networks.
Prado-Prado FJ, Martinez de la Vega O, Uriarte E, Ubeira FM, Chou KC, González-Díaz H.
Bioorg Med Chem (2009) 17 : 569 -575
PubMed 19112024 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 6.78 9.77

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL674 OSELTAMIVIR CARBOXYLATE -1.0 1 9.77
CHEMBL221722 FAVIPIRAVIR 4.0 1 7.32
CHEMBL222813 ZANAMIVIR 4.0 1 6.12
CHEMBL1229 OSELTAMIVIR 4.0 1 5.84
CHEMBL1643 RIBAVIRIN 4.0 1 4.86

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL674 OSELTAMIVIR CARBOXYLATE IC50 = 0.17 nM 9.77
CHEMBL221722 FAVIPIRAVIR IC50 = 48.0 nM 7.32
CHEMBL222813 ZANAMIVIR IC50 = 760.0 nM 6.12
CHEMBL1229 OSELTAMIVIR IC50 = 1450.0 nM 5.84
CHEMBL1643 RIBAVIRIN IC50 = 13800.0 nM 4.86