Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL1036445

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of human recombinant DNMT3b2
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

DNA (cytosine-5)-methyltransferase 3B (CHEMBL6095)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Constrained (l-)-S-adenosyl-l-homocysteine (SAH) analogues as DNA methyltransferase inhibitors.
Isakovic L, Saavedra OM, Llewellyn DB, Claridge S, Zhan L, Bernstein N, Vaisburg A, Elowe N, Petschner AJ, Rahil J, Beaulieu N, Gauthier F, MacLeod AR, Delorme D, Besterman JM, Wahhab A.
Bioorg Med Chem Lett (2009) 19 : 2742 -2746
PubMed 19364644 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 21 5.09 6.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL418052 S-ADENOSYLHOMOCYSTEINE 1 6.70
CHEMBL555257 1 6.58
CHEMBL557902 1 6.52
CHEMBL559283 1 6.04
CHEMBL550440 1 5.82
CHEMBL560106 1 5.72
CHEMBL558883 1 4.96
CHEMBL564052 1 4.92
CHEMBL538693 1 4.77
CHEMBL562689 1 4.68
CHEMBL551100 1 4.58
CHEMBL560768 1 4.57
CHEMBL551174 1 4.48
CHEMBL551787 1 4.41
CHEMBL563938 1 4.39
CHEMBL563230 1 4.27
CHEMBL559281 1 4.18
CHEMBL563782 1 4.00
CHEMBL539449 1 -
CHEMBL563888 1 -
CHEMBL538627 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL418052 S-ADENOSYLHOMOCYSTEINE IC50 = 200.0 nM 6.70
CHEMBL555257 IC50 = 260.0 nM 6.58
CHEMBL557902 IC50 = 300.0 nM 6.52
CHEMBL559283 IC50 = 920.0 nM 6.04
CHEMBL550440 IC50 = 1500.0 nM 5.82
CHEMBL560106 IC50 = 1900.0 nM 5.72
CHEMBL558883 IC50 = 11000.0 nM 4.96
CHEMBL564052 IC50 = 12000.0 nM 4.92
CHEMBL538693 IC50 = 17000.0 nM 4.77
CHEMBL562689 IC50 = 21000.0 nM 4.68
CHEMBL551100 IC50 = 26000.0 nM 4.58
CHEMBL560768 IC50 = 27000.0 nM 4.57
CHEMBL551174 IC50 = 33000.0 nM 4.48
CHEMBL551787 IC50 = 39000.0 nM 4.41
CHEMBL563938 IC50 = 41000.0 nM 4.39
CHEMBL563230 IC50 = 54000.0 nM 4.27
CHEMBL559281 IC50 = 66000.0 nM 4.18
CHEMBL563782 IC50 = 100000.0 nM 4.00
CHEMBL539449 IC50 > 100000.0 nM -
CHEMBL563888 IC50 > 100000.0 nM -
CHEMBL538627 IC50 > 45000.0 nM -