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Assay Detail

CHEMBL1040901

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human U87 cells after 72 hrs by trypan blue exclusion assay
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type U-87MG ATCC
Confidence 1 — Organism
Curated By Autocuration

Publication

Synthesis of new alkylaminooxysterols with potent cell differentiating activities: identification of leads for the treatment of cancer and neurodegenerative diseases.
de Medina P, Paillasse MR, Payré B, Silvente-Poirot S, Poirot M.
J Med Chem (2009) 52 : 7765 -7777
PubMed 19821610 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Activity 1 - -
IC50 1 6.13 6.13

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL567015 DENDROGENIN A 1 6.13
CHEMBL566588 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL567015 DENDROGENIN A IC50 = 740.0 nM 6.13
CHEMBL566588 Activity - -