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Assay Detail

CHEMBL1045382

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Functional
Antiviral activity against Vaccinia virus Lederle infected in HEL cells assessed as inhibition of virus-induced cytopathicity in presence of vildagliptin
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Vaccinia virus
Cell Type HEL
Confidence 1 — Organism
Curated By Autocuration

Target

Vaccinia virus (CHEMBL613493)
Type ORGANISM
Organism Vaccinia virus

Publication

Application of the dipeptidyl peptidase IV (DPPIV/CD26) based prodrug approach to different amine-containing drugs.
Diez-Torrubia A, García-Aparicio C, Cabrera S, De Meester I, Balzarini J, Camarasa MJ, Velázquez S.
J Med Chem (2010) 53 : 559 -572
PubMed 20000418 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 5.00 5.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1090 VIDARABINE 4.0 1 5.00
CHEMBL572009 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1090 VIDARABINE EC50 = 10000.0 nM 5.00
CHEMBL572009 EC50 = 135000.0 nM -