Assay Detail

CHEMBL1047439

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Functional

Antitrypanosomal activity against Trypanosoma brucei rhodesiense

ChEMBL ↗

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Target

Trypanosoma brucei rhodesiense (CHEMBL612348) ↗

Open DB target context

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Trypanosoma brucei rhodesiense (CHEMBL612348) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target Trypanosoma brucei rhodesiense

CHEMBL612348

Anchored from Assay target.

Protein identity Trypanosoma brucei rhodesiense

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Functional
Organism	Trypanosoma brucei rhodesiense
Confidence	1 — Organism
Curated By	Autocuration

Target

Trypanosoma brucei rhodesiense (CHEMBL612348) ↗

Type	ORGANISM
Organism	Trypanosoma brucei rhodesiense

Publication

Neglected tropical diseases: multi-target-directed ligands in the search for novel lead candidates against Trypanosoma and Leishmania.

Cavalli A, Bolognesi ML.
J Med Chem (2009) 52 : 7339 -7359
PubMed 19606868 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
IC50	1	7.10	7.10

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL256155	—	—	1	7.10

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL256155	—	IC50	=	80.0	nM	7.10