Assay Detail
Binding
CHEMBL1050880
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]WIN-55212-2 from CB1 receptor in rat cerebellar membrane after 90 mins by scintillation counting
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Tissue | Cerebellum |
| Subcellular | Membrane |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
Synthesis and pharmacological evaluation of sulfamide-based analogues of anandamide.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 5.37 | 5.37 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL374746 | — | — | 1 | 5.37 |
| CHEMBL219156 | — | — | 1 | - |
| CHEMBL437157 | — | — | 1 | - |
| CHEMBL218643 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL374746 | — | Ki | = | 4229.0 | nM | 5.37 |
| CHEMBL219156 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL437157 | — | Ki | > | 100000.0 | nM | - |
| CHEMBL218643 | — | Ki | > | 10000.0 | nM | - |