Assay Detail
Binding
CHEMBL1066432
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Competitive-type inhibition of autotaxin-mediated FS3 hydrolysis by Michaelis-Menten analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Characterization of non-lipid autotaxin inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 5.51 | 5.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL268789 | — | — | 1 | 5.72 |
| CHEMBL442472 | — | — | 1 | 5.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL268789 | — | Ki | = | 1900.0 | nM | 5.72 |
| CHEMBL442472 | — | Ki | = | 5000.0 | nM | 5.30 |