Assay Detail
Binding
CHEMBL1101970
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity to rat brain CB2 receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Radiosynthesis of novel carbon-11-labeled triaryl ligands for cannabinoid-type 2 receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.10 | 9.57 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1076680 | — | — | 1 | 9.57 |
| CHEMBL1081609 | — | — | 1 | 8.63 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1076680 | — | Ki | = | 0.27 | nM | 9.57 |
| CHEMBL1081609 | — | Ki | = | 2.32 | nM | 8.63 |