Assay Detail
Binding
CHEMBL1104415
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity at 5HT1A receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
The development and validation of a novel virtual screening cascade protocol to identify potential serotonin 5-HT(7)R antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.77 | 8.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1091933 | — | — | 1 | 8.10 |
| CHEMBL1094908 | — | — | 1 | 7.44 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1091933 | — | Ki | = | 8.0 | nM | 8.10 |
| CHEMBL1094908 | — | Ki | = | 36.0 | nM | 7.44 |