Assay Detail
ADMET
CHEMBL1104541
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Cytotoxicity against mouse NIH/3T3 cells assessed as viable cells after 72 hrs by MTT assay
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Mus musculus |
| Cell Type | NIH3T3 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Investigating the anti-proliferative activity of styrylazanaphthalenes and azanaphthalenediones.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 17 | 5.69 | 5.93 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1090672 | — | — | 1 | 5.93 |
| CHEMBL47360 | — | — | 1 | 5.62 |
| CHEMBL1089792 | — | — | 1 | 5.52 |
| CHEMBL1091870 | — | — | 1 | - |
| CHEMBL1092203 | — | — | 1 | - |
| CHEMBL1092204 | — | — | 1 | - |
| CHEMBL1092205 | — | — | 1 | - |
| CHEMBL1092206 | — | — | 1 | - |
| CHEMBL1091869 | — | — | 1 | - |
| CHEMBL1091029 | — | — | 1 | - |
| CHEMBL1089789 | — | — | 1 | - |
| CHEMBL1089790 | — | — | 1 | - |
| CHEMBL1089791 | — | — | 1 | - |
| CHEMBL1093129 | — | — | 1 | - |
| CHEMBL1093130 | — | — | 1 | - |
| CHEMBL241908 | — | — | 1 | - |
| CHEMBL1091028 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1090672 | — | IC50 | = | 1170.0 | nM | 5.93 |
| CHEMBL47360 | — | IC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL1089792 | — | IC50 | = | 3040.0 | nM | 5.52 |
| CHEMBL1091870 | — | IC50 | - | — | - | |
| CHEMBL1092203 | — | IC50 | - | — | - | |
| CHEMBL1092204 | — | IC50 | - | — | - | |
| CHEMBL1092205 | — | IC50 | - | — | - | |
| CHEMBL1092206 | — | IC50 | - | — | - | |
| CHEMBL1091869 | — | IC50 | - | — | - | |
| CHEMBL1091029 | — | IC50 | - | — | - | |
| CHEMBL1089789 | — | IC50 | - | — | - | |
| CHEMBL1089790 | — | IC50 | - | — | - | |
| CHEMBL1089791 | — | IC50 | - | — | - | |
| CHEMBL1093129 | — | IC50 | - | — | - | |
| CHEMBL1093130 | — | IC50 | - | — | - | |
| CHEMBL241908 | — | IC50 | - | — | - | |
| CHEMBL1091028 | — | IC50 | - | — | - |