Assay Detail
Functional
CHEMBL1105508
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at recombinant GluA4 receptor flop isoform expressed in Xenopus oocytes
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | Oocyte |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 5.09 | 5.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL602962 | — | — | 1 | 5.77 |
| CHEMBL575060 | GLUTAMIC ACID | 3.0 | 1 | 5.09 |
| CHEMBL73698 | — | — | 1 | 4.41 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL602962 | — | EC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL575060 | GLUTAMIC ACID | EC50 | = | 8100.0 | nM | 5.09 |
| CHEMBL73698 | — | EC50 | = | 39000.0 | nM | 4.41 |