Assay Detail
Binding
CHEMBL1106174
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of Acinetobacter baumannii beta-lactamase OXA40
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Acinetobacter baumannii |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
4,7-Dichloro benzothien-2-yl sulfonylaminomethyl boronic acid: first boronic acid-derived beta-lactamase inhibitor with class A, C, and D activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.25 | 5.25 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1089781 | — | — | 1 | 5.25 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1089781 | — | IC50 | = | 5600.0 | nM | 5.25 |