Assay Detail

CHEMBL1107396

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional

Agonist activity at P2Y receptor by [35S]GTPgammaS binding assay

ChEMBL ↗

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Target

Unchecked (CHEMBL612545) ↗

Open DB target context

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Unchecked (CHEMBL612545) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target Unchecked

CHEMBL612545

Anchored from Assay target.

Protein identity Unchecked

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Functional
Confidence	0 — Uncurated / Unknown
Curated By	Autocuration

Target

Unchecked (CHEMBL612545) ↗

Type

UNCHECKED

Publication

Frontal affinity chromatography-mass spectrometry useful for characterization of new ligands for GPR17 receptor.

Calleri E, Ceruti S, Cristalli G, Martini C, Temporini C, Parravicini C, Volpini R, Daniele S, Caccialanza G, Lecca D, Lambertucci C, Trincavelli ML, Marucci G, Wainer IW, Ranghino G, Fantucci P, Abbracchio MP, Massolini G.
J Med Chem (2010) 53 : 3489 -3501
PubMed 20394377 · DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
EC50	1	5.94	5.94

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL1096401	UDP TRISODIUM	—	1	5.94

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL1096401	UDP TRISODIUM	EC50	=	1140.0	nM	5.94