Assay Detail
Functional
CHEMBL1107472
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Inhibition of LTB4-stimulated human neutrophils migration after 30 mins by using CyQuant GR fluorescent dye
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Neutrophil |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery of novel and potent leukotriene B4 receptor antagonists. Part 1.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 9.12 | 10.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1098560 | — | — | 1 | 10.00 |
| CHEMBL1094346 | — | — | 1 | 10.00 |
| CHEMBL1099331 | — | — | 1 | 9.70 |
| CHEMBL1099335 | — | — | 1 | 9.70 |
| CHEMBL1094347 | — | — | 1 | 9.70 |
| CHEMBL1099337 | — | — | 1 | 9.15 |
| CHEMBL1099330 | — | — | 1 | 8.74 |
| CHEMBL1094348 | — | — | 1 | 8.43 |
| CHEMBL1094349 | — | — | 1 | 8.12 |
| CHEMBL1099334 | — | — | 1 | 7.70 |
| CHEMBL1099332 | — | — | 1 | - |
| CHEMBL1099333 | — | — | 1 | - |
| CHEMBL1099336 | — | — | 1 | - |
| CHEMBL1099338 | — | — | 1 | - |
| CHEMBL1094350 | — | — | 1 | - |
| CHEMBL15766 | LY-255283 | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1098560 | — | IC50 | = | 0.1 | nM | 10.00 |
| CHEMBL1094346 | — | IC50 | = | 0.1 | nM | 10.00 |
| CHEMBL1099331 | — | IC50 | = | 0.2 | nM | 9.70 |
| CHEMBL1099335 | — | IC50 | = | 0.2 | nM | 9.70 |
| CHEMBL1094347 | — | IC50 | = | 0.2 | nM | 9.70 |
| CHEMBL1099337 | — | IC50 | = | 0.7 | nM | 9.15 |
| CHEMBL1099330 | — | IC50 | = | 1.8 | nM | 8.74 |
| CHEMBL1094348 | — | IC50 | = | 3.68 | nM | 8.43 |
| CHEMBL1094349 | — | IC50 | = | 7.67 | nM | 8.12 |
| CHEMBL1099334 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL1099332 | — | IC50 | - | — | - | |
| CHEMBL1099333 | — | IC50 | - | — | - | |
| CHEMBL1099336 | — | IC50 | - | — | - | |
| CHEMBL1099338 | — | IC50 | - | — | - | |
| CHEMBL1094350 | — | IC50 | - | — | - | |
| CHEMBL15766 | LY-255283 | IC50 | - | — | - |