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Assay Detail

CHEMBL1107720

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Cytotoxicity against human CCRF-CEM cells after 48 hrs by MTT assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type CCRF-CEM
Confidence 1 — Organism
Curated By Autocuration

Target

CCRF-CEM (CHEMBL382)
Type CELL-LINE
Organism Homo sapiens

Publication

Structure and cytotoxicity of arnamial and related fungal sesquiterpene aryl esters.
Misiek M, Williams J, Schmich K, Hüttel W, Merfort I, Salomon CE, Aldrich CC, Hoffmeister D.
J Nat Prod (2009) 72 : 1888 -1891
PubMed 19795841 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 4.57 5.05

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1078389 ARNAMIAL 1 5.05
CHEMBL1078144 MELLEDONAL C 1 4.83
CHEMBL1078142 MELLEOLIDE D 1 4.21
CHEMBL1077563 1 4.20

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1078389 ARNAMIAL IC50 = 8910.0 nM 5.05
CHEMBL1078144 MELLEDONAL C IC50 = 14750.0 nM 4.83
CHEMBL1078142 MELLEOLIDE D IC50 = 61660.0 nM 4.21
CHEMBL1077563 IC50 = 63230.0 nM 4.20