Assay Detail
Binding
CHEMBL1108123
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Activity at human recombinant GluA2 flop isoform expressed in HEK203 cells assessed as blocked of receptor desensitization
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | HEK203 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Developing a complete pharmacology for AMPA receptors: a perspective on subtype-selective ligands.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 5.84 | 5.84 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1097939 | — | — | 1 | 5.84 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1097939 | — | EC50 | = | 1440.0 | nM | 5.84 |