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Assay Detail

CHEMBL1115016

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Herpes simplex virus 2 G infected in HEL cells assessed as protection from virus-induced cytopathogenicity after 2 to 3 days by MTT assay
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human alphaherpesvirus 2
Cell Type HEL
Confidence 1 — Organism
Curated By Autocuration

Target

Human alphaherpesvirus 2 (CHEMBL370)
Type ORGANISM
Organism Human alphaherpesvirus 2

Publication

Synthesis, antibacterial and antiviral properties of curcumin bioconjugates bearing dipeptide, fatty acids and folic acid.
Singh RK, Rai D, Yadav D, Bhargava A, Balzarini J, De Clercq E.
Eur J Med Chem (2010) 45 : 1078 -1086
PubMed 20034711 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 9 6.03 8.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL140 CURCUMIN 3.0 1 8.00
CHEMBL182 GANCICLOVIR 4.0 1 7.52
CHEMBL31634 BRIVUDINE 2.0 1 4.30
CHEMBL1643 RIBAVIRIN 4.0 1 4.30
CHEMBL1077034 1 -
CHEMBL1077033 1 -
CHEMBL1077031 1 -
CHEMBL1077035 1 -
CHEMBL1077036 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL140 CURCUMIN EC50 = 10.0 nM 8.00
CHEMBL182 GANCICLOVIR EC50 = 30.0 nM 7.52
CHEMBL31634 BRIVUDINE EC50 = 50000.0 nM 4.30
CHEMBL1643 RIBAVIRIN EC50 = 50000.0 nM 4.30
CHEMBL1077034 EC50 > 38.0 nM -
CHEMBL1077033 EC50 > 147.0 nM -
CHEMBL1077031 EC50 > 82.0 nM -
CHEMBL1077035 EC50 > 11.0 nM -
CHEMBL1077036 EC50 > 119.0 nM -