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Assay Detail

CHEMBL1116293

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to androgen receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Androgen receptor (CHEMBL1871)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Imaging progesterone receptor in breast tumors: synthesis and receptor binding affinity of fluoroalkyl-substituted analogues of tanaproget.
Zhou HB, Lee JH, Mayne CG, Carlson KE, Katzenellenbogen JA.
J Med Chem (2010) 53 : 3349 -3360
PubMed 20355713 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 9.22 9.22

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL166444 METRIBOLONE 2.0 1 9.22

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL166444 METRIBOLONE Kd = 0.6 nM 9.22