Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL1120962

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of CRF1 receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Corticotropin-releasing factor receptor 1 (CHEMBL1800)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Lessons learned from herbal medicinal products: the example of St. John's Wort (perpendicular).
Nahrstedt A, Butterweck V.
J Nat Prod (2010) 73 : 1015 -1021
PubMed 20408551 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.52 6.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL286494 HYPERICIN 3.0 1 6.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL286494 HYPERICIN IC50 = 300.0 nM 6.52