Assay Detail
Functional
CHEMBL1175602
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Antitumor activity against mouse SW1 cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | SW1 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Synthesis and preliminary evaluation of neuroprotection of celastrol analogues in PC12 cells.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 6.52 | 6.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1170915 | — | — | 1 | 6.52 |
| CHEMBL54804 | PRISTIMERIN | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1170915 | — | EC50 | = | 300.0 | nM | 6.52 |
| CHEMBL54804 | PRISTIMERIN | EC50 | < | 100.0 | nM | - |