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Assay Detail

CHEMBL1217675

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Binding
Inhibition of tyrosinase
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Identification of a potent and noncytotoxic inhibitor of melanin production.
Hwang S, Choi SY, Lee JH, Kim S, In J, Ha SK, Lee E, Kim TY, Kim SY, Choi S, Kim S.
Bioorg Med Chem (2010) 18 : 5602 -5609
PubMed 20615711 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 4.67 5.21

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL287556 KOJIC ACID 1 5.21
CHEMBL537 HYDROQUINONE 4.0 1 4.12
CHEMBL232202 ARBUTIN 2.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL287556 KOJIC ACID IC50 = 6200.0 nM 5.21
CHEMBL537 HYDROQUINONE IC50 = 75000.0 nM 4.12
CHEMBL232202 ARBUTIN IC50 = 17000000.0 nM -