Assay Detail
Binding
CHEMBL1219852
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of beta-1 adrenoceptor ( assessed as residual activity at 1 uM )
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Identification of orally available naphthyridine protein kinase D inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.63 | 5.63 |
| Activity | 1 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1214998 | — | — | 1 | 5.63 |
| CHEMBL1214857 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1214998 | — | IC50 | = | 2351.0 | nM | 5.63 |
| CHEMBL1214857 | — | Activity | > | 10000.0 | nM | - |