Assay Detail
Binding
CHEMBL1249833
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Inhibition of CDK2/cyclinA at 10 mM
4
Total Activities
4
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 6 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Target
Cyclin-dependent kinase 2/cyclin A (CHEMBL2094128) ↗| Type | PROTEIN COMPLEX |
| Organism | Homo sapiens |
Publication
Pharmacological inhibitors of glycogen synthase kinase 3.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Inhibition | 2 | - | - |
| IC50 | 2 | 5.00 | 5.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL156987 | — | — | 1 | 5.00 |
| CHEMBL1242556 | — | — | 1 | - |
| CHEMBL407373 | — | — | 1 | - |
| CHEMBL326705 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL156987 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL1242556 | — | Inhibition | = | 90.0 | % | - |
| CHEMBL407373 | — | Inhibition | = | 95.0 | % | - |
| CHEMBL326705 | — | IC50 | = | 250000.0 | nM | - |