Assay Detail
Binding
CHEMBL1253142
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Displacement of [3H]-oxytocin from rat oxytocin receptor expressed in HEK293-EBNA cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Cell Type | HEK293-EBNA |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Oral oxytocin antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.17 | 9.17 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1254117 | — | — | 1 | 9.17 |
| CHEMBL445816 | — | — | 1 | 9.17 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1254117 | — | Ki | = | 0.67 | nM | 9.17 |
| CHEMBL445816 | — | Ki | = | 0.67 | nM | 9.17 |