Assay Detail
Binding
CHEMBL1274071
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Inhibition of bovine liver beta-glucosidase after 10 to 30 mins
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bos taurus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Fluorescent-tagged sp2-iminosugars with potent β-glucosidase inhibitory activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 5 | 4.72 | 5.43 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1271962 | — | — | 1 | 5.43 |
| CHEMBL1269789 | — | — | 1 | 4.64 |
| CHEMBL1272018 | — | — | 1 | 4.54 |
| CHEMBL1269790 | — | — | 1 | 4.50 |
| CHEMBL1272019 | — | — | 1 | 4.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1271962 | — | Ki | = | 3700.0 | nM | 5.43 |
| CHEMBL1269789 | — | Ki | = | 23000.0 | nM | 4.64 |
| CHEMBL1272018 | — | Ki | = | 29000.0 | nM | 4.54 |
| CHEMBL1269790 | — | Ki | = | 32000.0 | nM | 4.50 |
| CHEMBL1272019 | — | Ki | = | 32000.0 | nM | 4.50 |