Assay Detail
Binding
CHEMBL1287449
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Binding affinity to human adenosine A2A receptor
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Molecular modeling study on potent and selective adenosine A(3) receptor agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 5.75 | 6.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL375190 | — | — | 1 | 6.44 |
| CHEMBL1277040 | — | — | 1 | 5.75 |
| CHEMBL574597 | — | — | 1 | 5.07 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL375190 | — | Ki | = | 363.0 | nM | 6.44 |
| CHEMBL1277040 | — | Ki | = | 1760.0 | nM | 5.75 |
| CHEMBL574597 | — | Ki | = | 8530.0 | nM | 5.07 |