Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL1293136

Review assay metadata, readout intent, target linkage, and publication context from the same page.

ADMET
Cytotoxicity against human NFF after 96 hrs by sulforhodamine B assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type NFF
Confidence 1 — Organism
Curated By Autocuration

Target

NFF (CHEMBL614198)
Type CELL-LINE
Organism Homo sapiens

Publication

Antimalarial histone deacetylase inhibitors containing cinnamate or NSAID components.
Wheatley NC, Andrews KT, Tran TL, Lucke AJ, Reid RC, Fairlie DP.
Bioorg Med Chem Lett (2010) 20 : 7080 -7084
PubMed 20951583 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 6.53 6.77

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1289720 1 6.77
CHEMBL1289943 1 6.58
CHEMBL221654 1 6.24

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1289720 IC50 = 169.0 nM 6.77
CHEMBL1289943 IC50 = 260.0 nM 6.58
CHEMBL221654 IC50 = 570.0 nM 6.24