Assay Detail
Functional
CHEMBL1613869
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Luminescence Cell-Based Dose Response HTS to Identify Inhibitors of Luciferase Translation or Activity in H4 Neuroglioblastoma Cells. (Class of assay: confirmatory) [Related pubchem assays: 1813 (Primary HTS), 1827 (Project Summary)]
2032
Total Activities
2032
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2032 | 5.05 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1451921 | — | — | 1 | 7.00 |
| CHEMBL1491705 | — | — | 1 | 7.00 |
| CHEMBL1574553 | — | — | 1 | 6.97 |
| CHEMBL1423927 | — | — | 1 | 6.95 |
| CHEMBL2360527 | — | — | 1 | 6.95 |
| CHEMBL1333294 | — | — | 1 | 6.89 |
| CHEMBL1459841 | — | — | 1 | 6.89 |
| CHEMBL1488760 | — | — | 1 | 6.87 |
| CHEMBL65 | CAMPTOTHECIN | -1.0 | 1 | 6.87 |
| CHEMBL1570765 | — | — | 1 | 6.86 |
| CHEMBL1580848 | — | — | 1 | 6.85 |
| CHEMBL584458 | — | — | 1 | 6.85 |
| CHEMBL1332878 | — | — | 1 | 6.84 |
| CHEMBL1351441 | — | — | 1 | 6.84 |
| CHEMBL1349428 | — | — | 1 | 6.84 |
| CHEMBL3192140 | — | — | 1 | 6.84 |
| CHEMBL1537452 | — | — | 1 | 6.83 |
| CHEMBL1384292 | — | — | 1 | 6.80 |
| CHEMBL1329221 | — | — | 1 | 6.80 |
| CHEMBL3195189 | — | — | 1 | 6.77 |
| CHEMBL1986418 | — | — | 1 | 6.75 |
| CHEMBL1605021 | — | — | 1 | 6.71 |
| CHEMBL1491222 | — | — | 1 | 6.70 |
| CHEMBL1602637 | — | — | 1 | 6.70 |
| CHEMBL1334514 | — | — | 1 | 6.70 |
| CHEMBL3211308 | — | — | 1 | 6.68 |
| CHEMBL1525789 | — | — | 1 | 6.68 |
| CHEMBL1613639 | — | — | 1 | 6.67 |
| CHEMBL1468323 | — | — | 1 | 6.67 |
| CHEMBL600336 | — | — | 1 | 6.65 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1491705 | — | EC50 | = | 101.0 | nM | 7.00 |
| CHEMBL1451921 | — | EC50 | = | 101.0 | nM | 7.00 |
| CHEMBL1574553 | — | EC50 | = | 107.0 | nM | 6.97 |
| CHEMBL2360527 | — | EC50 | = | 112.0 | nM | 6.95 |
| CHEMBL1423927 | — | EC50 | = | 113.0 | nM | 6.95 |
| CHEMBL1333294 | — | EC50 | = | 129.0 | nM | 6.89 |
| CHEMBL1459841 | — | EC50 | = | 130.0 | nM | 6.89 |
| CHEMBL65 | CAMPTOTHECIN | EC50 | = | 134.0 | nM | 6.87 |
| CHEMBL1488760 | — | EC50 | = | 134.0 | nM | 6.87 |
| CHEMBL1570765 | — | EC50 | = | 137.0 | nM | 6.86 |
| CHEMBL584458 | — | EC50 | = | 142.0 | nM | 6.85 |
| CHEMBL1580848 | — | EC50 | = | 142.0 | nM | 6.85 |
| CHEMBL1351441 | — | EC50 | = | 143.0 | nM | 6.84 |
| CHEMBL1349428 | — | EC50 | = | 146.0 | nM | 6.84 |
| CHEMBL1332878 | — | EC50 | = | 146.0 | nM | 6.84 |
| CHEMBL3192140 | — | EC50 | = | 146.0 | nM | 6.84 |
| CHEMBL1537452 | — | EC50 | = | 148.0 | nM | 6.83 |
| CHEMBL1384292 | — | EC50 | = | 160.0 | nM | 6.80 |
| CHEMBL1329221 | — | EC50 | = | 158.0 | nM | 6.80 |
| CHEMBL3195189 | — | EC50 | = | 171.0 | nM | 6.77 |
| CHEMBL1986418 | — | EC50 | = | 178.0 | nM | 6.75 |
| CHEMBL1605021 | — | EC50 | = | 197.0 | nM | 6.71 |
| CHEMBL1334514 | — | EC50 | = | 201.0 | nM | 6.70 |
| CHEMBL1491222 | — | EC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1602637 | — | EC50 | = | 199.0 | nM | 6.70 |
| CHEMBL3211308 | — | EC50 | = | 208.0 | nM | 6.68 |
| CHEMBL1525789 | — | EC50 | = | 207.0 | nM | 6.68 |
| CHEMBL1613639 | — | EC50 | = | 216.0 | nM | 6.67 |
| CHEMBL1468323 | — | EC50 | = | 212.0 | nM | 6.67 |
| CHEMBL600336 | — | EC50 | = | 225.0 | nM | 6.65 |
| CHEMBL3195273 | — | EC50 | = | 229.0 | nM | 6.64 |
| CHEMBL601757 | — | EC50 | = | 235.0 | nM | 6.63 |
| CHEMBL1452795 | — | EC50 | = | 234.0 | nM | 6.63 |
| CHEMBL1864040 | — | EC50 | = | 239.0 | nM | 6.62 |
| CHEMBL290077 | — | EC50 | = | 242.0 | nM | 6.62 |
| CHEMBL1488730 | — | EC50 | = | 239.0 | nM | 6.62 |
| CHEMBL1352854 | — | EC50 | = | 238.0 | nM | 6.62 |
| CHEMBL1413629 | — | EC50 | = | 248.0 | nM | 6.61 |
| CHEMBL1998521 | — | EC50 | = | 244.0 | nM | 6.61 |
| CHEMBL1340058 | — | EC50 | = | 250.0 | nM | 6.60 |
| CHEMBL1581197 | — | EC50 | = | 251.0 | nM | 6.60 |
| CHEMBL1359872 | — | EC50 | = | 257.0 | nM | 6.59 |
| CHEMBL1497549 | — | EC50 | = | 266.0 | nM | 6.58 |
| CHEMBL1490339 | — | EC50 | = | 266.0 | nM | 6.58 |
| CHEMBL1459109 | — | EC50 | = | 269.0 | nM | 6.57 |
| CHEMBL1321622 | — | EC50 | = | 283.0 | nM | 6.55 |
| CHEMBL1990919 | — | EC50 | = | 292.0 | nM | 6.54 |
| CHEMBL1547760 | — | EC50 | = | 293.0 | nM | 6.53 |
| CHEMBL1256686 | CALCIMYCIN | EC50 | = | 293.0 | nM | 6.53 |
| CHEMBL1329237 | — | EC50 | = | 294.0 | nM | 6.53 |