Assay Detail
Functional
CHEMBL1613883
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Fluorescence-based counterscreen assay for S1P4 agonists: Cell-based dose response high throughput screening assay to identify agonists of the Sphingosine 1-Phosphate Receptor 1 (S1P1). (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1509, AID1523, AID1801, AID463107, AID463118, AID463119, AID463122, AID463123, AID463129, AID463225, AID504400, AID504460]
46
Total Activities
46
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 46 | 5.09 | 5.93 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3195883 | — | — | 1 | 5.93 |
| CHEMBL1409828 | — | — | 1 | 5.68 |
| CHEMBL1447076 | — | — | 1 | 5.66 |
| CHEMBL1577139 | — | — | 1 | 5.66 |
| CHEMBL46874 | PINAFIDE | 2.0 | 1 | 5.51 |
| CHEMBL1533401 | — | — | 1 | 5.51 |
| CHEMBL1467763 | — | — | 1 | 5.50 |
| CHEMBL153064 | — | — | 1 | 5.38 |
| CHEMBL1531320 | — | — | 1 | 5.30 |
| CHEMBL1375375 | — | — | 1 | 5.26 |
| CHEMBL1537907 | — | — | 1 | 5.22 |
| CHEMBL1442207 | — | — | 1 | 5.13 |
| CHEMBL1342332 | — | — | 1 | 5.10 |
| CHEMBL1341200 | — | — | 1 | 5.06 |
| CHEMBL1362307 | — | — | 1 | 5.00 |
| CHEMBL1375597 | — | — | 1 | 4.98 |
| CHEMBL1501839 | — | — | 1 | 4.97 |
| CHEMBL1605463 | — | — | 1 | 4.90 |
| CHEMBL1419836 | — | — | 1 | 4.80 |
| CHEMBL1402796 | — | — | 1 | 4.69 |
| CHEMBL1604216 | — | — | 1 | 4.66 |
| CHEMBL1300662 | — | — | 1 | 4.61 |
| CHEMBL1456255 | — | — | 1 | 4.47 |
| CHEMBL358644 | — | — | 1 | 4.28 |
| CHEMBL1993778 | — | — | 1 | 4.03 |
| CHEMBL1604434 | — | — | 1 | - |
| CHEMBL1363676 | — | — | 1 | - |
| CHEMBL1349615 | — | — | 1 | - |
| CHEMBL1539075 | — | — | 1 | - |
| CHEMBL1580856 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3195883 | — | EC50 | = | 1180.0 | nM | 5.93 |
| CHEMBL1409828 | — | EC50 | = | 2080.0 | nM | 5.68 |
| CHEMBL1577139 | — | EC50 | = | 2180.0 | nM | 5.66 |
| CHEMBL1447076 | — | EC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL46874 | PINAFIDE | EC50 | = | 3110.0 | nM | 5.51 |
| CHEMBL1533401 | — | EC50 | = | 3120.0 | nM | 5.51 |
| CHEMBL1467763 | — | EC50 | = | 3130.0 | nM | 5.50 |
| CHEMBL153064 | — | EC50 | = | 4140.0 | nM | 5.38 |
| CHEMBL1531320 | — | EC50 | = | 5050.0 | nM | 5.30 |
| CHEMBL1375375 | — | EC50 | = | 5450.0 | nM | 5.26 |
| CHEMBL1537907 | — | EC50 | = | 5980.0 | nM | 5.22 |
| CHEMBL1442207 | — | EC50 | = | 7490.0 | nM | 5.13 |
| CHEMBL1342332 | — | EC50 | = | 7880.0 | nM | 5.10 |
| CHEMBL1341200 | — | EC50 | = | 8750.0 | nM | 5.06 |
| CHEMBL1362307 | — | EC50 | = | 10100.0 | nM | 5.00 |
| CHEMBL1375597 | — | EC50 | = | 10400.0 | nM | 4.98 |
| CHEMBL1501839 | — | EC50 | = | 10600.0 | nM | 4.97 |
| CHEMBL1605463 | — | EC50 | = | 12500.0 | nM | 4.90 |
| CHEMBL1419836 | — | EC50 | = | 15900.0 | nM | 4.80 |
| CHEMBL1402796 | — | EC50 | = | 20400.0 | nM | 4.69 |
| CHEMBL1604216 | — | EC50 | = | 22000.0 | nM | 4.66 |
| CHEMBL1300662 | — | EC50 | = | 24600.0 | nM | 4.61 |
| CHEMBL1456255 | — | EC50 | = | 33500.0 | nM | 4.47 |
| CHEMBL358644 | — | EC50 | = | 52900.0 | nM | 4.28 |
| CHEMBL1993778 | — | EC50 | = | 93500.0 | nM | 4.03 |
| CHEMBL1427987 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1332070 | — | EC50 | > | 5530.0 | nM | - |
| CHEMBL1982477 | — | EC50 | > | 5530.0 | nM | - |
| CHEMBL1459145 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1377446 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1537481 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1351890 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1320243 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL3190474 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1319154 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1384911 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1503105 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1422092 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1607677 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1530797 | — | EC50 | > | 614.0 | nM | - |
| CHEMBL1562579 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1580856 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1539075 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1349615 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1363676 | — | EC50 | > | 49800.0 | nM | - |
| CHEMBL1604434 | — | EC50 | > | 49800.0 | nM | - |