Assay Detail
Functional
CHEMBL1613923
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: A cytotoxicity screen of small molecule inhibitors of the PhoP region in Salmonella typhi identified in the primary screen. (Class of assay: confirmatory) [Related pubchem assays: 1850, 1864, 1985 ]
1509
Total Activities
1504
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1509 | 5.00 | 6.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1521960 | — | — | 1 | 6.70 |
| CHEMBL1481347 | — | — | 1 | 6.68 |
| CHEMBL1396209 | — | — | 1 | 6.66 |
| CHEMBL1499792 | — | — | 1 | 6.52 |
| CHEMBL727 | THIOGUANINE | 4.0 | 1 | 6.50 |
| CHEMBL290077 | — | — | 1 | 6.46 |
| CHEMBL1200883 | THONZONIUM BROMIDE | 4.0 | 1 | 6.44 |
| CHEMBL1977877 | — | — | 1 | 6.44 |
| CHEMBL1373096 | — | — | 1 | 6.44 |
| CHEMBL3199665 | — | — | 1 | 6.42 |
| CHEMBL1996730 | — | — | 1 | 6.38 |
| CHEMBL461579 | — | — | 1 | 6.36 |
| CHEMBL1382884 | — | — | 1 | 6.36 |
| CHEMBL1332756 | — | — | 1 | 6.33 |
| CHEMBL1375045 | — | — | 1 | 6.32 |
| CHEMBL1335846 | — | — | 1 | 6.31 |
| CHEMBL1596681 | — | — | 1 | 6.28 |
| CHEMBL3189405 | — | — | 1 | 6.24 |
| CHEMBL589670 | — | — | 1 | 6.21 |
| CHEMBL242580 | CICLOPIROX OLAMINE | 3.0 | 1 | 6.20 |
| CHEMBL586135 | — | — | 1 | 6.19 |
| CHEMBL1437516 | — | — | 1 | 6.18 |
| CHEMBL1450086 | — | — | 1 | 6.17 |
| CHEMBL1524986 | — | — | 1 | 6.16 |
| CHEMBL1587596 | — | — | 1 | 6.15 |
| CHEMBL1242180 | — | — | 1 | 6.15 |
| CHEMBL405110 | METHYLENE BLUE ANHYDROUS | 4.0 | 1 | 6.14 |
| CHEMBL466853 | — | — | 1 | 6.14 |
| CHEMBL1448592 | — | — | 1 | 6.13 |
| CHEMBL1546374 | — | — | 1 | 6.12 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1521960 | — | EC50 | = | 200.0 | nM | 6.70 |
| CHEMBL1481347 | — | EC50 | = | 210.0 | nM | 6.68 |
| CHEMBL1396209 | — | EC50 | = | 220.0 | nM | 6.66 |
| CHEMBL1499792 | — | EC50 | = | 300.0 | nM | 6.52 |
| CHEMBL727 | THIOGUANINE | EC50 | = | 320.0 | nM | 6.50 |
| CHEMBL290077 | — | EC50 | = | 350.0 | nM | 6.46 |
| CHEMBL1200883 | THONZONIUM BROMIDE | EC50 | = | 360.0 | nM | 6.44 |
| CHEMBL1373096 | — | EC50 | = | 360.0 | nM | 6.44 |
| CHEMBL1977877 | — | EC50 | = | 360.0 | nM | 6.44 |
| CHEMBL3199665 | — | EC50 | = | 380.0 | nM | 6.42 |
| CHEMBL1996730 | — | EC50 | = | 420.0 | nM | 6.38 |
| CHEMBL1382884 | — | EC50 | = | 440.0 | nM | 6.36 |
| CHEMBL461579 | — | EC50 | = | 440.0 | nM | 6.36 |
| CHEMBL1332756 | — | EC50 | = | 470.0 | nM | 6.33 |
| CHEMBL1375045 | — | EC50 | = | 480.0 | nM | 6.32 |
| CHEMBL1335846 | — | EC50 | = | 490.0 | nM | 6.31 |
| CHEMBL1596681 | — | EC50 | = | 520.0 | nM | 6.28 |
| CHEMBL3189405 | — | EC50 | = | 570.0 | nM | 6.24 |
| CHEMBL589670 | — | EC50 | = | 620.0 | nM | 6.21 |
| CHEMBL242580 | CICLOPIROX OLAMINE | EC50 | = | 630.0 | nM | 6.20 |
| CHEMBL586135 | — | EC50 | = | 650.0 | nM | 6.19 |
| CHEMBL1437516 | — | EC50 | = | 660.0 | nM | 6.18 |
| CHEMBL1450086 | — | EC50 | = | 680.0 | nM | 6.17 |
| CHEMBL1524986 | — | EC50 | = | 700.0 | nM | 6.16 |
| CHEMBL1242180 | — | EC50 | = | 710.0 | nM | 6.15 |
| CHEMBL1587596 | — | EC50 | = | 710.0 | nM | 6.15 |
| CHEMBL466853 | — | EC50 | = | 720.0 | nM | 6.14 |
| CHEMBL405110 | METHYLENE BLUE ANHYDROUS | EC50 | = | 720.0 | nM | 6.14 |
| CHEMBL1448592 | — | EC50 | = | 740.0 | nM | 6.13 |
| CHEMBL1546374 | — | EC50 | = | 760.0 | nM | 6.12 |
| CHEMBL1347071 | — | EC50 | = | 820.0 | nM | 6.09 |
| CHEMBL1487183 | ALEXIDINE HYDROCHLORIDE | EC50 | = | 830.0 | nM | 6.08 |
| CHEMBL1304363 | — | EC50 | = | 840.0 | nM | 6.08 |
| CHEMBL1987461 | — | EC50 | = | 900.0 | nM | 6.05 |
| CHEMBL1363219 | — | EC50 | = | 900.0 | nM | 6.05 |
| CHEMBL3192432 | — | EC50 | = | 970.0 | nM | 6.01 |
| CHEMBL1423463 | — | EC50 | = | 970.0 | nM | 6.01 |
| CHEMBL3193098 | — | EC50 | = | 990.0 | nM | 6.00 |
| CHEMBL1306460 | — | EC50 | = | 1010.0 | nM | 6.00 |
| CHEMBL581868 | — | EC50 | = | 1050.0 | nM | 5.98 |
| CHEMBL1420037 | — | EC50 | = | 1050.0 | nM | 5.98 |
| CHEMBL1321398 | — | EC50 | = | 1180.0 | nM | 5.93 |
| CHEMBL548615 | — | EC50 | = | 1190.0 | nM | 5.92 |
| CHEMBL428064 | — | EC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL1544371 | — | EC50 | = | 1240.0 | nM | 5.91 |
| CHEMBL1349146 | — | EC50 | = | 1270.0 | nM | 5.90 |
| CHEMBL1569910 | — | EC50 | = | 1250.0 | nM | 5.90 |
| CHEMBL1370471 | — | EC50 | = | 1290.0 | nM | 5.89 |
| CHEMBL2359911 | — | EC50 | = | 1290.0 | nM | 5.89 |
| CHEMBL532849 | — | EC50 | = | 1360.0 | nM | 5.87 |