Assay Detail
Functional
CHEMBL1613951
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: BAP1 Enzyme inhibitors Dose Response Confirmation. (Class of assay: confirmatory) [Related pubchem assays: 436 (Primary screen preceding this dose response confirmation assay.)]
42
Total Activities
42
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Ubiquitin carboxyl-terminal hydrolase BAP1 (CHEMBL1293314) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 42 | 4.61 | 5.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1548217 | — | — | 1 | 5.05 |
| CHEMBL1307842 | — | — | 1 | 4.98 |
| CHEMBL1419387 | — | — | 1 | 4.86 |
| CHEMBL1609890 | — | — | 1 | 4.76 |
| CHEMBL1563909 | — | — | 1 | 4.74 |
| CHEMBL1462119 | — | — | 1 | 4.73 |
| CHEMBL1527746 | — | — | 1 | 4.69 |
| CHEMBL3189877 | — | — | 1 | 4.65 |
| CHEMBL1330121 | — | — | 1 | 4.64 |
| CHEMBL1460841 | — | — | 1 | 4.63 |
| CHEMBL1427879 | — | — | 1 | 4.63 |
| CHEMBL1413198 | — | — | 1 | 4.54 |
| CHEMBL1535453 | — | — | 1 | 4.52 |
| CHEMBL1347594 | — | — | 1 | 4.52 |
| CHEMBL3190584 | — | — | 1 | 4.47 |
| CHEMBL1611354 | — | — | 1 | 4.45 |
| CHEMBL1407201 | — | — | 1 | 4.44 |
| CHEMBL1471212 | — | — | 1 | 4.43 |
| CHEMBL1535124 | — | — | 1 | 4.41 |
| CHEMBL1410132 | — | — | 1 | 4.38 |
| CHEMBL1528716 | — | — | 1 | 4.35 |
| CHEMBL1541809 | — | — | 1 | - |
| CHEMBL1425173 | — | — | 1 | - |
| CHEMBL1528655 | — | — | 1 | - |
| CHEMBL1529788 | — | — | 1 | - |
| CHEMBL1361464 | — | — | 1 | - |
| CHEMBL1469705 | — | — | 1 | - |
| CHEMBL1578559 | — | — | 1 | - |
| CHEMBL1451988 | — | — | 1 | - |
| CHEMBL1388979 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1548217 | — | IC50 | = | 9002.3 | nM | 5.05 |
| CHEMBL1307842 | — | IC50 | = | 10487.3 | nM | 4.98 |
| CHEMBL1419387 | — | IC50 | = | 13926.8 | nM | 4.86 |
| CHEMBL1609890 | — | IC50 | = | 17282.0 | nM | 4.76 |
| CHEMBL1563909 | — | IC50 | = | 18282.8 | nM | 4.74 |
| CHEMBL1462119 | — | IC50 | = | 18728.9 | nM | 4.73 |
| CHEMBL1527746 | — | IC50 | = | 20376.0 | nM | 4.69 |
| CHEMBL3189877 | — | IC50 | = | 22562.5 | nM | 4.65 |
| CHEMBL1330121 | — | IC50 | = | 23100.9 | nM | 4.64 |
| CHEMBL1460841 | — | IC50 | = | 23373.1 | nM | 4.63 |
| CHEMBL1427879 | — | IC50 | = | 23329.7 | nM | 4.63 |
| CHEMBL1413198 | — | IC50 | = | 29128.0 | nM | 4.54 |
| CHEMBL1535453 | — | IC50 | = | 30229.7 | nM | 4.52 |
| CHEMBL1347594 | — | IC50 | = | 30395.3 | nM | 4.52 |
| CHEMBL3190584 | — | IC50 | = | 33938.6 | nM | 4.47 |
| CHEMBL1611354 | — | IC50 | = | 35796.2 | nM | 4.45 |
| CHEMBL1407201 | — | IC50 | = | 36623.5 | nM | 4.44 |
| CHEMBL1471212 | — | IC50 | = | 36743.5 | nM | 4.43 |
| CHEMBL1535124 | — | IC50 | = | 38559.0 | nM | 4.41 |
| CHEMBL1410132 | — | IC50 | = | 41626.7 | nM | 4.38 |
| CHEMBL1528716 | — | IC50 | = | 44797.8 | nM | 4.35 |
| CHEMBL1560511 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1437943 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1455209 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1543947 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1540610 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1383713 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1607205 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1522605 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1347985 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1322572 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1440883 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1601197 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1388979 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1451988 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1578559 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1469705 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1361464 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1529788 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1528655 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1425173 | — | IC50 | > | 50000.0 | nM | - |
| CHEMBL1541809 | — | IC50 | > | 50000.0 | nM | - |