Assay Detail
Functional
CHEMBL1614012
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Dose response counterscreen for antagonists of galanin receptor 2 (GalR2): a cell-based high-throughput screening assay for inhibitors of beta-lactamase activity. (Class of assay: confirmatory) [Related pubchem assays: 828, 1225, 866 ]
47
Total Activities
47
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 47 | 4.88 | 5.12 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1447697 | — | — | 1 | 5.12 |
| CHEMBL1400481 | — | — | 1 | 5.02 |
| CHEMBL309016 | — | — | 1 | 4.96 |
| CHEMBL1458812 | — | — | 1 | 4.77 |
| CHEMBL1586531 | — | — | 1 | 4.77 |
| CHEMBL1374788 | — | — | 1 | 4.77 |
| CHEMBL1531933 | — | — | 1 | 4.75 |
| CHEMBL1428566 | — | — | 1 | - |
| CHEMBL1567331 | — | — | 1 | - |
| CHEMBL1418247 | — | — | 1 | - |
| CHEMBL1585420 | — | — | 1 | - |
| CHEMBL1452324 | — | — | 1 | - |
| CHEMBL1352348 | — | — | 1 | - |
| CHEMBL1432794 | — | — | 1 | - |
| CHEMBL1353474 | — | — | 1 | - |
| CHEMBL1342746 | — | — | 1 | - |
| CHEMBL1330152 | — | — | 1 | - |
| CHEMBL1242180 | — | — | 1 | - |
| CHEMBL1427917 | — | — | 1 | - |
| CHEMBL1372292 | — | — | 1 | - |
| CHEMBL1347469 | — | — | 1 | - |
| CHEMBL1582794 | — | — | 1 | - |
| CHEMBL1573112 | — | — | 1 | - |
| CHEMBL1534042 | — | — | 1 | - |
| CHEMBL1482215 | — | — | 1 | - |
| CHEMBL1403484 | — | — | 1 | - |
| CHEMBL578515 | — | — | 1 | - |
| CHEMBL1598827 | — | — | 1 | - |
| CHEMBL1463624 | — | — | 1 | - |
| CHEMBL1466965 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1447697 | — | IC50 | = | 7528.0 | nM | 5.12 |
| CHEMBL1400481 | — | IC50 | = | 9608.0 | nM | 5.02 |
| CHEMBL309016 | — | IC50 | = | 11080.0 | nM | 4.96 |
| CHEMBL1458812 | — | IC50 | = | 17070.0 | nM | 4.77 |
| CHEMBL1586531 | — | IC50 | = | 16970.0 | nM | 4.77 |
| CHEMBL1374788 | — | IC50 | = | 17100.0 | nM | 4.77 |
| CHEMBL1531933 | — | IC50 | = | 17900.0 | nM | 4.75 |
| CHEMBL1401057 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1330152 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1566205 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1320867 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1320669 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1499501 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1360480 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1567331 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1242180 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1438200 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1451772 | — | IC50 | > | 14000.0 | nM | - |
| CHEMBL415879 | PHENANTHROLINE | IC50 | > | 42000.0 | nM | - |
| CHEMBL116569 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1382898 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1423004 | — | IC50 | = | 2529000.0 | nM | - |
| CHEMBL1540377 | — | IC50 | > | 14000.0 | nM | - |
| CHEMBL1462076 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1570553 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1362352 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1987060 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1347469 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1466965 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1463624 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1598827 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL578515 | — | IC50 | > | 14000.0 | nM | - |
| CHEMBL1403484 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1482215 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1534042 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1573112 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1582794 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1342746 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1372292 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1427917 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1428566 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1418247 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1585420 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1452324 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1352348 | — | IC50 | > | 42000.0 | nM | - |
| CHEMBL1432794 | — | IC50 | > | 14000.0 | nM | - |
| CHEMBL1353474 | — | IC50 | > | 42000.0 | nM | - |