Assay Detail
Functional
CHEMBL1614030
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: HTS dose response assay for identification of inhibitors of TNFa-specific NF-kB induction. (Class of assay: confirmatory) [Related pubchem assays (depositor defined):AID1566, AID1575, AID1578, AID1579, AID1852, AID2337]
546
Total Activities
546
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Category | confirmatory |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 546 | 5.25 | 6.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1507251 | — | — | 1 | 6.46 |
| CHEMBL1580556 | — | — | 1 | 6.35 |
| CHEMBL1351908 | — | — | 1 | 6.32 |
| CHEMBL1480238 | — | — | 1 | 6.18 |
| CHEMBL3210725 | — | — | 1 | 6.15 |
| CHEMBL1507713 | — | — | 1 | 6.13 |
| CHEMBL1361922 | — | — | 1 | 6.11 |
| CHEMBL1427335 | — | — | 1 | 6.08 |
| CHEMBL1415184 | — | — | 1 | 6.04 |
| CHEMBL1505956 | — | — | 1 | 6.02 |
| CHEMBL1319304 | — | — | 1 | 6.01 |
| CHEMBL1520241 | — | — | 1 | 5.98 |
| CHEMBL3194944 | — | — | 1 | 5.95 |
| CHEMBL1887153 | — | — | 1 | 5.93 |
| CHEMBL1313090 | — | — | 1 | 5.92 |
| CHEMBL1351128 | — | — | 1 | 5.92 |
| CHEMBL190346 | — | — | 1 | 5.90 |
| CHEMBL1466636 | — | — | 1 | 5.89 |
| CHEMBL1505474 | — | — | 1 | 5.85 |
| CHEMBL3195189 | — | — | 1 | 5.85 |
| CHEMBL1361883 | — | — | 1 | 5.82 |
| CHEMBL1538692 | — | — | 1 | 5.82 |
| CHEMBL1416848 | — | — | 1 | 5.81 |
| CHEMBL1465720 | — | — | 1 | 5.79 |
| CHEMBL1337226 | — | — | 1 | 5.79 |
| CHEMBL1332684 | — | — | 1 | 5.79 |
| CHEMBL1550862 | — | — | 1 | 5.79 |
| CHEMBL1583186 | — | — | 1 | 5.78 |
| CHEMBL1372398 | — | — | 1 | 5.77 |
| CHEMBL1305930 | — | — | 1 | 5.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1507251 | — | IC50 | = | 344.75 | nM | 6.46 |
| CHEMBL1580556 | — | IC50 | = | 451.0 | nM | 6.35 |
| CHEMBL1351908 | — | IC50 | = | 477.75 | nM | 6.32 |
| CHEMBL1480238 | — | IC50 | = | 666.25 | nM | 6.18 |
| CHEMBL3210725 | — | IC50 | = | 702.75 | nM | 6.15 |
| CHEMBL1507713 | — | IC50 | = | 748.5 | nM | 6.13 |
| CHEMBL1361922 | — | IC50 | = | 783.25 | nM | 6.11 |
| CHEMBL1427335 | — | IC50 | = | 841.75 | nM | 6.08 |
| CHEMBL1415184 | — | IC50 | = | 921.5 | nM | 6.04 |
| CHEMBL1505956 | — | IC50 | = | 949.5 | nM | 6.02 |
| CHEMBL1319304 | — | IC50 | = | 970.5 | nM | 6.01 |
| CHEMBL1520241 | — | IC50 | = | 1046.0 | nM | 5.98 |
| CHEMBL3194944 | — | IC50 | = | 1133.5 | nM | 5.95 |
| CHEMBL1887153 | — | IC50 | = | 1161.0 | nM | 5.93 |
| CHEMBL1313090 | — | IC50 | = | 1194.0 | nM | 5.92 |
| CHEMBL1351128 | — | IC50 | = | 1207.0 | nM | 5.92 |
| CHEMBL190346 | — | IC50 | = | 1270.5 | nM | 5.90 |
| CHEMBL1466636 | — | IC50 | = | 1288.5 | nM | 5.89 |
| CHEMBL3195189 | — | IC50 | = | 1404.25 | nM | 5.85 |
| CHEMBL1505474 | — | IC50 | = | 1422.5 | nM | 5.85 |
| CHEMBL1538692 | — | IC50 | = | 1511.0 | nM | 5.82 |
| CHEMBL1361883 | — | IC50 | = | 1526.0 | nM | 5.82 |
| CHEMBL1416848 | — | IC50 | = | 1539.5 | nM | 5.81 |
| CHEMBL1465720 | — | IC50 | = | 1606.0 | nM | 5.79 |
| CHEMBL1337226 | — | IC50 | = | 1615.5 | nM | 5.79 |
| CHEMBL1332684 | — | IC50 | = | 1610.0 | nM | 5.79 |
| CHEMBL1550862 | — | IC50 | = | 1628.0 | nM | 5.79 |
| CHEMBL1583186 | — | IC50 | = | 1678.0 | nM | 5.78 |
| CHEMBL1305930 | — | IC50 | = | 1708.0 | nM | 5.77 |
| CHEMBL1372398 | — | IC50 | = | 1715.0 | nM | 5.77 |
| CHEMBL1565526 | — | IC50 | = | 1730.0 | nM | 5.76 |
| CHEMBL3196263 | — | IC50 | = | 1765.75 | nM | 5.75 |
| CHEMBL1540477 | — | IC50 | = | 1836.5 | nM | 5.74 |
| CHEMBL1455542 | — | IC50 | = | 1832.0 | nM | 5.74 |
| CHEMBL1486619 | — | IC50 | = | 1809.0 | nM | 5.74 |
| CHEMBL1379291 | — | IC50 | = | 1826.0 | nM | 5.74 |
| CHEMBL1386754 | — | IC50 | = | 1827.5 | nM | 5.74 |
| CHEMBL3195322 | — | IC50 | = | 1824.75 | nM | 5.74 |
| CHEMBL1324011 | — | IC50 | = | 1889.0 | nM | 5.72 |
| CHEMBL585502 | — | IC50 | = | 1901.5 | nM | 5.72 |
| CHEMBL1376861 | — | IC50 | = | 1903.5 | nM | 5.72 |
| CHEMBL578257 | — | IC50 | = | 1957.5 | nM | 5.71 |
| CHEMBL1504069 | — | IC50 | = | 1940.5 | nM | 5.71 |
| CHEMBL1300239 | — | IC50 | = | 1932.0 | nM | 5.71 |
| CHEMBL1364018 | — | IC50 | = | 2106.5 | nM | 5.68 |
| CHEMBL1568646 | — | IC50 | = | 2067.5 | nM | 5.68 |
| CHEMBL1610725 | — | IC50 | = | 2102.5 | nM | 5.68 |
| CHEMBL1612423 | — | IC50 | = | 2111.0 | nM | 5.68 |
| CHEMBL3189810 | — | IC50 | = | 2130.5 | nM | 5.67 |
| CHEMBL1375966 | — | IC50 | = | 2120.0 | nM | 5.67 |