Assay Detail
Functional
CHEMBL1614071
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: Counterscreen for IDE inhibitors: Luminescence-based cell-based high throughput dose response assay to identify compounds that are cytotoxic to HEK cells. (Class of assay: confirmatory) [Related pubchem assays: 434962 (Primary screen (IDE inhibitors in singlicate)), 449730 (Counterscreen (Cytotoxicity in triplicate)), 435028 (Confirmation (IDE inhibitors in triplicate)), 434984 (Summary (IDE inhibitors))]
127
Total Activities
127
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | HEK293 |
| Category | confirmatory |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 127 | 4.69 | 8.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1364530 | — | — | 1 | 8.41 |
| CHEMBL1423690 | — | — | 1 | 4.98 |
| CHEMBL1371792 | — | — | 1 | 4.96 |
| CHEMBL1487402 | — | — | 1 | 4.95 |
| CHEMBL1570108 | — | — | 1 | 4.94 |
| CHEMBL1596609 | — | — | 1 | 4.92 |
| CHEMBL1995565 | — | — | 1 | 4.88 |
| CHEMBL1569711 | — | — | 1 | 4.87 |
| CHEMBL1557186 | — | — | 1 | 4.85 |
| CHEMBL1369585 | — | — | 1 | 4.84 |
| CHEMBL1363026 | — | — | 1 | 4.84 |
| CHEMBL393287 | — | — | 1 | 4.84 |
| CHEMBL597857 | — | — | 1 | 4.84 |
| CHEMBL1559626 | — | — | 1 | 4.81 |
| CHEMBL2001792 | — | — | 1 | 4.80 |
| CHEMBL1366556 | — | — | 1 | 4.80 |
| CHEMBL1489113 | — | — | 1 | 4.80 |
| CHEMBL1978101 | — | — | 1 | 4.79 |
| CHEMBL1420311 | — | — | 1 | 4.78 |
| CHEMBL1596457 | — | — | 1 | 4.78 |
| CHEMBL1981990 | — | — | 1 | 4.78 |
| CHEMBL1349451 | — | — | 1 | 4.77 |
| CHEMBL1414359 | — | — | 1 | 4.76 |
| CHEMBL1425837 | — | — | 1 | 4.76 |
| CHEMBL1382246 | — | — | 1 | 4.75 |
| CHEMBL1377807 | — | — | 1 | 4.74 |
| CHEMBL372629 | — | — | 1 | 4.74 |
| CHEMBL1445779 | — | — | 1 | 4.74 |
| CHEMBL1469797 | — | — | 1 | 4.72 |
| CHEMBL1458192 | — | — | 1 | 4.71 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1364530 | — | IC50 | = | 3.9 | nM | 8.41 |
| CHEMBL1423690 | — | IC50 | = | 10474.0 | nM | 4.98 |
| CHEMBL1371792 | — | IC50 | = | 10972.0 | nM | 4.96 |
| CHEMBL1487402 | — | IC50 | = | 11137.0 | nM | 4.95 |
| CHEMBL1570108 | — | IC50 | = | 11575.0 | nM | 4.94 |
| CHEMBL1596609 | — | IC50 | = | 12056.0 | nM | 4.92 |
| CHEMBL1995565 | — | IC50 | = | 13069.0 | nM | 4.88 |
| CHEMBL1569711 | — | IC50 | = | 13562.0 | nM | 4.87 |
| CHEMBL1557186 | — | IC50 | = | 14041.0 | nM | 4.85 |
| CHEMBL1363026 | — | IC50 | = | 14402.0 | nM | 4.84 |
| CHEMBL597857 | — | IC50 | = | 14276.0 | nM | 4.84 |
| CHEMBL1369585 | — | IC50 | = | 14467.0 | nM | 4.84 |
| CHEMBL393287 | — | IC50 | = | 14379.0 | nM | 4.84 |
| CHEMBL1559626 | — | IC50 | = | 15470.0 | nM | 4.81 |
| CHEMBL1489113 | — | IC50 | = | 15864.0 | nM | 4.80 |
| CHEMBL1366556 | — | IC50 | = | 15736.0 | nM | 4.80 |
| CHEMBL2001792 | — | IC50 | = | 16002.0 | nM | 4.80 |
| CHEMBL1978101 | — | IC50 | = | 16284.0 | nM | 4.79 |
| CHEMBL1981990 | — | IC50 | = | 16557.0 | nM | 4.78 |
| CHEMBL1420311 | — | IC50 | = | 16512.0 | nM | 4.78 |
| CHEMBL1596457 | — | IC50 | = | 16545.0 | nM | 4.78 |
| CHEMBL1349451 | — | IC50 | = | 17126.0 | nM | 4.77 |
| CHEMBL1425837 | — | IC50 | = | 17538.0 | nM | 4.76 |
| CHEMBL1414359 | — | IC50 | = | 17396.0 | nM | 4.76 |
| CHEMBL1382246 | — | IC50 | = | 17591.0 | nM | 4.75 |
| CHEMBL1445779 | — | IC50 | = | 18211.0 | nM | 4.74 |
| CHEMBL1377807 | — | IC50 | = | 18408.0 | nM | 4.74 |
| CHEMBL372629 | — | IC50 | = | 18110.0 | nM | 4.74 |
| CHEMBL1469797 | — | IC50 | = | 19000.0 | nM | 4.72 |
| CHEMBL1458192 | — | IC50 | = | 19396.0 | nM | 4.71 |
| CHEMBL1375130 | — | IC50 | = | 19315.0 | nM | 4.71 |
| CHEMBL1450467 | — | IC50 | = | 19327.0 | nM | 4.71 |
| CHEMBL1309068 | — | IC50 | = | 19400.0 | nM | 4.71 |
| CHEMBL3189228 | — | IC50 | = | 20008.0 | nM | 4.70 |
| CHEMBL1549566 | — | IC50 | = | 19820.0 | nM | 4.70 |
| CHEMBL1598813 | — | IC50 | = | 20843.0 | nM | 4.68 |
| CHEMBL1366394 | — | IC50 | = | 20710.0 | nM | 4.68 |
| CHEMBL117121 | — | IC50 | = | 21188.0 | nM | 4.67 |
| CHEMBL1499996 | — | IC50 | = | 21179.0 | nM | 4.67 |
| CHEMBL1424237 | — | IC50 | = | 22056.0 | nM | 4.66 |
| CHEMBL1526622 | — | IC50 | = | 22456.0 | nM | 4.65 |
| CHEMBL1483950 | — | IC50 | = | 22557.0 | nM | 4.65 |
| CHEMBL1538650 | — | IC50 | = | 22317.0 | nM | 4.65 |
| CHEMBL1483555 | — | IC50 | = | 22399.0 | nM | 4.65 |
| CHEMBL1344703 | — | IC50 | = | 22400.0 | nM | 4.65 |
| CHEMBL1342644 | — | IC50 | = | 23043.0 | nM | 4.64 |
| CHEMBL1469359 | — | IC50 | = | 22918.0 | nM | 4.64 |
| CHEMBL1451796 | — | IC50 | = | 23811.0 | nM | 4.62 |
| CHEMBL1410800 | — | IC50 | = | 23848.0 | nM | 4.62 |
| CHEMBL1388661 | — | IC50 | = | 24760.0 | nM | 4.61 |