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Assay Detail

CHEMBL1614183

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
PUBCHEM_BIOASSAY: High Throughput Screen to Identify Inhibitors of Mycobacterium tuberculosis H37Rv. (Class of assay: confirmatory)
2044
Total Activities
2044
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Category confirmatory
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

PubChem BioAssay data set

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2044 5.43 6.71

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1557648 1 6.71
CHEMBL3145126 1 6.71
CHEMBL1493936 1 6.71
CHEMBL1503257 1 6.71
CHEMBL1488980 1 6.71
CHEMBL1415310 1 6.71
CHEMBL1532755 1 6.71
CHEMBL1481301 1 6.71
CHEMBL1598279 1 6.71
CHEMBL1402807 1 6.71
CHEMBL1580472 1 6.71
CHEMBL1580076 1 6.71
CHEMBL1501506 1 6.71
CHEMBL1461196 1 6.71
CHEMBL1539205 1 6.71
CHEMBL1497418 1 6.71
CHEMBL1539109 1 6.71
CHEMBL1372421 1 6.71
CHEMBL1332111 1 6.71
CHEMBL306946 TRYPTANTHRIN 1 6.71
CHEMBL1993431 1 6.71
CHEMBL3191258 1 6.71
CHEMBL1528219 1 6.71
CHEMBL548615 1 6.71
CHEMBL1300641 1 6.71
CHEMBL597871 1 6.71
CHEMBL1498307 1 6.71
CHEMBL1537522 1 6.71
CHEMBL1576330 1 6.71
CHEMBL1605089 1 6.71

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1542886 IC50 = 195.0 nM 6.71
CHEMBL1587645 IC50 = 195.0 nM 6.71
CHEMBL1550564 IC50 = 195.0 nM 6.71
CHEMBL1598279 IC50 = 195.0 nM 6.71
CHEMBL1481301 IC50 = 195.0 nM 6.71
CHEMBL597871 IC50 = 195.0 nM 6.71
CHEMBL1415310 IC50 = 195.0 nM 6.71
CHEMBL1488980 IC50 = 195.0 nM 6.71
CHEMBL548615 IC50 = 195.0 nM 6.71
CHEMBL1532755 IC50 = 195.0 nM 6.71
CHEMBL1503257 IC50 = 195.0 nM 6.71
CHEMBL1509475 IC50 = 195.0 nM 6.71
CHEMBL1557648 IC50 = 195.0 nM 6.71
CHEMBL1461196 IC50 = 195.0 nM 6.71
CHEMBL3145126 IC50 = 195.0 nM 6.71
CHEMBL1528219 IC50 = 195.0 nM 6.71
CHEMBL1425667 IC50 = 195.0 nM 6.71
CHEMBL1521482 IC50 = 195.0 nM 6.71
CHEMBL1539205 IC50 = 195.0 nM 6.71
CHEMBL1300641 IC50 = 195.0 nM 6.71
CHEMBL1539109 IC50 = 195.0 nM 6.71
CHEMBL1406270 IC50 = 195.0 nM 6.71
CHEMBL1546739 IC50 = 195.0 nM 6.71
CHEMBL1493936 IC50 = 195.0 nM 6.71
CHEMBL1390275 IC50 = 195.0 nM 6.71
CHEMBL1501506 IC50 = 195.0 nM 6.71
CHEMBL1471716 IC50 = 195.0 nM 6.71
CHEMBL1537522 IC50 = 195.0 nM 6.71
CHEMBL1483676 IC50 = 195.0 nM 6.71
CHEMBL1427858 IC50 = 195.0 nM 6.71
CHEMBL306946 TRYPTANTHRIN IC50 = 195.0 nM 6.71
CHEMBL1498307 IC50 = 195.0 nM 6.71
CHEMBL1367268 IC50 = 195.0 nM 6.71
CHEMBL1332111 IC50 = 195.0 nM 6.71
CHEMBL1993431 IC50 = 195.0 nM 6.71
CHEMBL1576330 IC50 = 195.0 nM 6.71
CHEMBL1313101 IC50 = 195.0 nM 6.71
CHEMBL1580076 IC50 = 195.0 nM 6.71
CHEMBL1497418 IC50 = 195.0 nM 6.71
CHEMBL3191258 IC50 = 195.0 nM 6.71
CHEMBL1547352 IC50 = 195.0 nM 6.71
CHEMBL1561287 IC50 = 195.0 nM 6.71
CHEMBL3190733 IC50 = 195.0 nM 6.71
CHEMBL1372421 IC50 = 195.0 nM 6.71
CHEMBL1584777 IC50 = 195.0 nM 6.71
CHEMBL1580472 IC50 = 195.0 nM 6.71
CHEMBL1349073 EFLOXATE IC50 = 195.0 nM 6.71
CHEMBL1404109 IC50 = 195.0 nM 6.71
CHEMBL1402807 IC50 = 195.0 nM 6.71
CHEMBL1605089 IC50 = 195.0 nM 6.71