Assay Detail
Binding
CHEMBL1614255
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PUBCHEM_BIOASSAY: HTS identification of compounds inhibiting phosphomannose isomerase (PMI) via a fluorescence intensity assay. (Class of assay: confirmatory) [Related pubchem assays: 1220 ]
191
Total Activities
191
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Category | confirmatory |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
PubChem BioAssay data set
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 191 | 4.86 | 5.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1392651 | — | — | 1 | 5.89 |
| CHEMBL1310318 | — | — | 1 | 5.54 |
| CHEMBL175266 | — | — | 1 | 5.45 |
| CHEMBL1489071 | — | — | 1 | 5.42 |
| CHEMBL1438240 | — | — | 1 | 5.41 |
| CHEMBL1432427 | — | — | 1 | 5.39 |
| CHEMBL1390710 | — | — | 1 | 5.37 |
| CHEMBL3191714 | — | — | 1 | 5.35 |
| CHEMBL75913 | — | — | 1 | 5.32 |
| CHEMBL1465693 | — | — | 1 | 5.29 |
| CHEMBL1339149 | — | — | 1 | 5.28 |
| CHEMBL1995112 | — | — | 1 | 5.27 |
| CHEMBL1550861 | — | — | 1 | 5.22 |
| CHEMBL3196976 | — | — | 1 | 5.18 |
| CHEMBL1336959 | — | — | 1 | 5.17 |
| CHEMBL1400481 | — | — | 1 | 5.16 |
| CHEMBL3191022 | — | — | 1 | 5.15 |
| CHEMBL1374283 | — | — | 1 | 5.14 |
| CHEMBL1453636 | — | — | 1 | 5.13 |
| CHEMBL1527869 | — | — | 1 | 5.08 |
| CHEMBL1602859 | — | — | 1 | 5.07 |
| CHEMBL1608601 | — | — | 1 | 5.07 |
| CHEMBL1422255 | — | — | 1 | 5.03 |
| CHEMBL1417290 | — | — | 1 | 5.00 |
| CHEMBL3193349 | — | — | 1 | 4.99 |
| CHEMBL1369932 | — | — | 1 | 4.96 |
| CHEMBL1910223 | — | — | 1 | 4.96 |
| CHEMBL1589626 | — | — | 1 | 4.96 |
| CHEMBL1605045 | — | — | 1 | 4.95 |
| CHEMBL1571704 | — | — | 1 | 4.95 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1392651 | — | IC50 | = | 1272.9 | nM | 5.89 |
| CHEMBL1310318 | — | IC50 | = | 2905.4 | nM | 5.54 |
| CHEMBL175266 | — | IC50 | = | 3550.0 | nM | 5.45 |
| CHEMBL1489071 | — | IC50 | = | 3786.6 | nM | 5.42 |
| CHEMBL1438240 | — | IC50 | = | 3927.9 | nM | 5.41 |
| CHEMBL1432427 | — | IC50 | = | 4087.8 | nM | 5.39 |
| CHEMBL1390710 | — | IC50 | = | 4299.9 | nM | 5.37 |
| CHEMBL3191714 | — | IC50 | = | 4500.9 | nM | 5.35 |
| CHEMBL75913 | — | IC50 | = | 4757.0 | nM | 5.32 |
| CHEMBL1465693 | — | IC50 | = | 5123.5 | nM | 5.29 |
| CHEMBL1339149 | — | IC50 | = | 5250.1 | nM | 5.28 |
| CHEMBL1995112 | — | IC50 | = | 5361.1 | nM | 5.27 |
| CHEMBL1550861 | — | IC50 | = | 6084.2 | nM | 5.22 |
| CHEMBL3196976 | — | IC50 | = | 6612.4 | nM | 5.18 |
| CHEMBL1336959 | — | IC50 | = | 6777.3 | nM | 5.17 |
| CHEMBL1400481 | — | IC50 | = | 6924.9 | nM | 5.16 |
| CHEMBL3191022 | — | IC50 | = | 7018.9 | nM | 5.15 |
| CHEMBL1374283 | — | IC50 | = | 7291.8 | nM | 5.14 |
| CHEMBL1453636 | — | IC50 | = | 7395.3 | nM | 5.13 |
| CHEMBL1527869 | — | IC50 | = | 8325.0 | nM | 5.08 |
| CHEMBL1608601 | — | IC50 | = | 8551.0 | nM | 5.07 |
| CHEMBL1602859 | — | IC50 | = | 8427.7 | nM | 5.07 |
| CHEMBL1422255 | — | IC50 | = | 9411.5 | nM | 5.03 |
| CHEMBL1417290 | — | IC50 | = | 10017.0 | nM | 5.00 |
| CHEMBL3193349 | — | IC50 | = | 10257.0 | nM | 4.99 |
| CHEMBL1369932 | — | IC50 | = | 10848.0 | nM | 4.96 |
| CHEMBL1910223 | — | IC50 | = | 11018.0 | nM | 4.96 |
| CHEMBL1589626 | — | IC50 | = | 10933.0 | nM | 4.96 |
| CHEMBL608699 | — | IC50 | = | 11223.0 | nM | 4.95 |
| CHEMBL1605045 | — | IC50 | = | 11181.0 | nM | 4.95 |
| CHEMBL1571704 | — | IC50 | = | 11117.0 | nM | 4.95 |
| CHEMBL1991599 | — | IC50 | = | 11573.0 | nM | 4.94 |
| CHEMBL1347373 | — | IC50 | = | 11703.0 | nM | 4.93 |
| CHEMBL1985664 | — | IC50 | = | 12011.0 | nM | 4.92 |
| CHEMBL1562260 | — | IC50 | = | 12667.0 | nM | 4.90 |
| CHEMBL1559622 | — | IC50 | = | 12547.0 | nM | 4.90 |
| CHEMBL1496326 | — | IC50 | = | 13694.0 | nM | 4.86 |
| CHEMBL1546522 | — | IC50 | = | 14160.0 | nM | 4.85 |
| CHEMBL75412 | — | IC50 | = | 14354.0 | nM | 4.84 |
| CHEMBL1374860 | — | IC50 | = | 14351.0 | nM | 4.84 |
| CHEMBL1334768 | — | IC50 | = | 14492.0 | nM | 4.84 |
| CHEMBL1499658 | — | IC50 | = | 15579.0 | nM | 4.81 |
| CHEMBL3198496 | — | IC50 | = | 15510.0 | nM | 4.81 |
| CHEMBL1329850 | — | IC50 | = | 16041.0 | nM | 4.79 |
| CHEMBL1478652 | — | IC50 | = | 16378.0 | nM | 4.79 |
| CHEMBL1550366 | — | IC50 | = | 16694.0 | nM | 4.78 |
| CHEMBL3196067 | — | IC50 | = | 18343.0 | nM | 4.74 |
| CHEMBL3192684 | — | IC50 | = | 19053.0 | nM | 4.72 |
| CHEMBL3197242 | — | IC50 | = | 19574.0 | nM | 4.71 |
| CHEMBL33027 | — | IC50 | = | 21303.0 | nM | 4.67 |